GPCR Modulation of Thieno[2,3-b]pyridine Anti-Proliferative Agents
نویسندگان
چکیده
منابع مشابه
GPCR Modulation of Thieno[2,3-b]pyridine Anti-Proliferative Agents.
A panel of docking scaffolds was developed for the known molecular targets of the anticancer agents, thieno[2,3-b]pyridines, in order to glean insight into their mechanism of action. The reported targets are the copper-trafficking antioxidant 1 protein, tyrosyl DNA phosphodiesterase 1, the colchicine binding site in tubulin, adenosine A2A receptor, and, finally, phospholipase C-δ1. According to...
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ژورنال
عنوان ژورنال: Molecules
سال: 2017
ISSN: 1420-3049
DOI: 10.3390/molecules22122254